Scopinal Tablets / Film-coated
Hyoscine Butyl Bromide
              10mg  
              
              Julphar (Gulf Pharmaceutical Industries)
                  
              
              | Pack size | 1000's (20's Blister x 50) | 
|---|---|
| Dispensing mode | POM | 
| Source | UAE | 
| Agent | JULPHAR | 
| Retail Price | 231.00 AED | 
Available as:
Indications
Scopinal Tablets / Film-coated is used for: 
 Gastrointestinal tract spasm, Abdominal pain, Genitourinary spasm
                                              
                        Adult Dose
Oral
Gastrointestinal tract spasm; Genitourinary spasm
Adult: 20 mg 4 times daily.
Parenteral
Gastrointestinal tract spasm; Genitourinary spasm
Adult: 20 mg IM/IV repeated after 30 min if needed.
Max Dosage: 100 mg daily.
                                              
                        Child Dose
Oral
Gastrointestinal tract spasm; Genitourinary spasm
Child: 6-12 yr: 10 mg tid.
                                              
                        Renal Dose
Administration
Contra Indications
Narrow-angle glaucoma, acute haemorrhage, paralytic ileus, tachycardia due to cardiac insufficiency, myasthenia gravis.
                                              
                        Precautions
Hepatic/renal disease, pyloric stenosis, urinary retention, prostatic hyperplasia, psychosis, seizure disorders, ulcerative colitis, coronary artery disease, tachyarrhythmias, heart failure, hypertension. Elderly, children, pregnancy, lactation.
                                              
                        Pregnancy-Lactation
Interactions
Additive sedative effects with alcohol or other CNS depressants. Reduced effects with acetylcholinesterase inhibitors (donepezil, galantamine, rivastigmine, tacrine).
Potentially Fatal: Effect potentiated by other anticholinergic drugs and TCAs.
                                              
                        Adverse Effects
Side effects of Hyoscine Butyl Bromide : 
 Flushing,  postural hypotension,  tachycardia,  fibrillation. Rarely psychotic reactions. Dizziness,  drowsiness,  fatigue,  headache,  memory loss. Dry skin,  erythema,  increased sensitivity to light,  rash. Bloatedness,  constipation,  dry throat,  dysphagia,  nausea,  vomiting,  xerostomia. Dysuria,  urinary retention. Tremor,  weakness. Impaired accommodation,  blurred vision,  cycloplegia,  dryness,  narrow-angle glaucoma,  increased intraocular pain,  itching,  photophobia,  pupil dilation. Dry nose. Decreased diaphoresis,  heat intolerance. Ophthalmic: Somnolence,  dermatitis,  oedema,  exudate,  follicular conjunctivitis,  increased IOP,  local irritation,  photophobia,  vascular and respiratory congestion.
Potentially Fatal: CNS depression,  coma,  circulatory and respiratory failure.
                                              
                        Mechanism of Action
Hyoscine competitively blocks muscarinic receptors and has central and peripheral actions. It relaxes smooth muscle and reduces gastric and intestinal motility.
                                              
                        Note
Scopinal 10mg Tablets / Film-coated manufactured by Julphar (Gulf Pharmaceutical Industries). Its generic name is Hyoscine Butyl Bromide. Scopinal is availble in United Arab Emirates.
 Farmaco UAE drug index information on Scopinal Tablets / Film-coated is not intended for diagnosis, medical advice or treatment; neither intended to be a substitute for the exercise of professional judgment.
                                        Some other brands of Hyoscine Butyl Bromide :
Injection
                        
                                Antipan
                                20mg/ml
                            
                            
                            
                                ARWAN PHARMACEUTICAL INDUSTRIES LEBANON s.a.l.
                            
                        Tablets
                        
                                Buscopan
                                10mg
                            
                            
                            
                                Boehringer Ingelheim GmbH
                            
                        Tablets / Sugar-coated
                        
                                Buscopan
                                10mg
                            
                            
                            
                                Boehringer Ingelheim International GmbH
                            
                        Tablets / Film-coated
                        
                                Hycom
                                10mg
                            
                            
                            
                                National Pharmaceutical industries Co. (SAOG)
                            
                        Tablets / Film-coated
                        
                                Hycom
                                10mg
                            
                            
                            
                                National Pharmaceutical industries Co. (SAOG)